Pitstop 1
CAS No. 1332879-51-2
Pitstop 1 ( Pitstop-1;Pitstop1 )
产品货号. M11323 CAS No. 1332879-51-2
A potent, selective inhibitor of clathrin-independent endocytosis with IC50 of 18 uM.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥7857 | 有现货 |
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50MG | ¥16038 | 有现货 |
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100MG | ¥20250 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Pitstop 1
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述A potent, selective inhibitor of clathrin-independent endocytosis with IC50 of 18 uM.
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产品描述A potent, selective inhibitor of clathrin-independent endocytosis with IC50 of 18 uM (inhibition of clathrin TD-amphiphysin B/C complex formation); inhibits endocytic recycling of synaptic vesicles in neurons and in situ.
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同义词Pitstop-1;Pitstop1
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通路Others
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靶点Clathrin
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受体Clathrin
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研究领域——
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适应症——
化学信息
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CAS Number1332879-51-2
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分子量404.37
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分子式C19H13N2NaO5S
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纯度>98% (HPLC)
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溶解度——
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SMILESNC1=CC=C(CN2C(C3=CC(S(=O)(O[Na])=O)=CC4=C3C(C2=O)=CC=C4)=O)C=C1
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化学全称2-(4-Aminobenzyl)-1,3-dioxo-2,3-dihydro-1H-benzo[de]isoquinoline-5-sulfonic acid sodium salt
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. von Kleist L, et al. Cell. 2011 Aug 5;146(3):471-84.
2. Nilewski LG, et al. ACS Chem Neurosci. 2017 Aug 14. doi: 10.1021/acschemneuro.7b00138.
2. Nilewski LG, et al. ACS Chem Neurosci. 2017 Aug 14. doi: 10.1021/acschemneuro.7b00138.
产品手册
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Pitstop 2 (b)
A small molecule inhibitor of clathrin terminal domain and inhibits clathrin-mediated endocytosis.
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Pitstop 1
A potent, selective inhibitor of clathrin-independent endocytosis with IC50 of 18 uM.